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Title of Journal: Amino Acids

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Abbravation: Amino Acids

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Springer Vienna

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1438-2199

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Analogues of both Leu and Metenkephalin containi

Authors: Roberta Galeazzi Gianluca Martelli Eleonora Marcucci Mario Orena Samuele Rinaldi Roberta Lattanzi Lucia Negri
Publish Date: 2009/07/08
Volume: 38, Issue: 4, Pages: 1057-1065
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Abstract

An efficient route was developed for the synthesis of the Fmocprotected dipeptide 4 isostere of GlyGly containing an αmethylene βamino acid the conformationally restricted analogues of Leuenkephalin 3a and Metenkephalin 3b respectively were prepared by changing 4 for Gly2Gly3 in the native compounds 3a and 3b whose biological activities were significantly lower than the parent compounds


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  6. Tissue-specific responses to loss of transglutaminase 2
  7. Regulation of intestinal protein metabolism by amino acids
  8. Free amino acid production during tomato fruit ripening: a focus on l -glutamate
  9. Bacterial signaling and adaptation
  10. Gas chromatographic determination and mechanism of formation of D-amino acids occurring in fermented and roasted cocoa beans, cocoa powder, chocolate and cocoa shell
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  13. Near infrared spectroscopy compared to liquid chromatography coupled to mass spectrometry and capillary electrophoresis as a detection tool for peptide reaction monitoring
  14. EPR spin-trapping of protein radicals to investigate biological oxidative mechanisms
  15. Kinetic study of racemization of aspartyl residues in synthetic elastin peptides
  16. Proteomics analysis of sensitive and tolerant barley genotypes under drought stress
  17. Camphoric acid stimulates osteoblast differentiation and induces glutamate receptor expression
  18. Taurine-like GABA aminotransferase inhibitors prevent rabbit brain slices against oxygen–glucose deprivation-induced damage
  19. Cardiovascular actions of l -cysteine and l -cysteine sulfinic acid in the nucleus tractus solitarius of the rat
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  23. Circular dichroism and cross-linking studies of bacteriorhodopsin mutants
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